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Cyclophosphamide
intestinal
transporter
Solute carrier
family 22
member 1
Canalicular
multispecific
organic anion
transporter 2
Acrylic acid
transporter
Phosphoramide
aziridinium
transporter
Alcophosphamide
transporter
4-Glutathionyl
cyclophosphamide
transporter
Nornitrogen
mustard
transporter
3-
Dechloroethylifosfamide
transporter
Chloroacetaldehyde
transporter
4-
Ketocyclophosphamide
transporter
Phosphoramide
mustard
transporter
Carboxyphosphamide
transporter
Cytochrome P450
2C9
Cytochrome P450
3A4
Cytochrome P450
3A7
Unknown
Aldehyde
dehydrogenase,
dimeric
NADP-preferring
Glutathione
S-transferase
A1
Alcohol
dehydrogenase
1A
Unknown
Unknown
Unknown
Aldehyde
dehydrogenase,
dimeric
NADP-preferring
Cyclophosphamide
4-Glutathionyl
cyclophosphamide
Chloroacetaldehyde
3-
Dechloroethylifosfamide
4-
Ketocyclophosphamide
Nornitrogen
mustard
Carboxyphosphamide
Alcophosphamide
Acrylic acid
Phosphoramide
Aziridinium
Phosphoramide
mustard
Cyclophosphamide
Cyclophosphamide
Cyclophosphamide
Cyclophosphamide
Cyclophosphamide
Cyclophosphamide
Aldophosphamide
Aldophosphamide
Acrylic acid
Phosphoramide
Aziridinium
Alcophosphamide
4-Glutathionyl
cyclophosphamide
Nornitrogen
mustard
3-
Dechloroethylifosfamide
Chloroacetaldehyde
4-
Ketocyclophosphamide
Phosphoramide
mustard
Carboxyphosphamide
O2
NADPH
H+
4-
Hydroxycyclophosphamide
H2 O
NADP
O2
H2 O
H2 O2
NAD
NADH
NAD
H2 O
NADH
H+
Glutathione
H2 O
NAD
NADH
H+
Acrolein
Cl-
NAD
H2 O
NADH
H+
Heme
Heme
Heme
Zinc
Excretion
Cytosol
Hepatocyte
Endoplasmic Reticulum
Intestinal Epithelial Cell
Endoplasmic Reticulum
Unknown
SLC22A1
ABCC3
Unknown
Unknown
Unknown
Unknown
Unknown
Unknown
Unknown
Unknown
Unknown
Unknown
CYP2C9
CYP3A4
CYP3A7
Unknown
ALDH3A1
GSTA1
ADH1A
Unknown
Unknown
Unknown
ALDH3A1
Cyclophosphamide
4-Glutathionyl
cyclophosphamide
Chloroacetaldehyde
3-
Dechloroethylifosfamide
4-
Ketocyclophosphamide
Nornitrogen
mustard
Carboxyphosphamide
Alcophosphamide
Acrylic acid
Phosphoramide
Aziridinium
Phosphoramide
mustard
Cyclophosphamide
Cyclophosphamide
Cyclophosphamide
Cyclophosphamide
Cyclophosphamide
Cyclophosphamide
Aldophosphamide
Aldophosphamide
Acrylic acid
Phosphoramide
Aziridinium
Alcophosphamide
4-Glutathionyl
cyclophosphamide
Nornitrogen
mustard
3-
Dechloroethylifosfamide
Chloroacetaldehyde
4-
Ketocyclophosphamide
Phosphoramide
mustard
Carboxyphosphamide
Oxygen
NADPH
Hydrogen Ion
4-
Hydroxycyclophosphamide
Water
NADP
Oxygen
Water
Hydrogen
peroxide
NAD
NADH
NAD
Water
NADH
Hydrogen Ion
Glutathione
Water
NAD
NADH
Hydrogen Ion
Acrolein
Chloride ion
NAD
Water
NADH
Hydrogen Ion
Excretion
SLC22A1
ABCC3
CYP2C9
CYP3A4
CYP3A7
ALDH3A1
GSTA1
ADH1A
ALDH3A1
Cycloph
4GtyCP
chlogl
3DCLFA
4KcycPm
Nornm
Caroxyp
Alcopho
AcryliA
PhoAzdm
Phospho
Cycloph
Cycloph
Cycloph
Cycloph
Cycloph
Cycloph
Aldoph
Aldoph
AcryliA
PhoAzdm
Alcopho
4GtyCP
Nornm
3DCLFA
chlogl
4KcycPm
Phospho
Caroxyp
O2
NADPH
H+
4HCP
H2 O
NADP
O2
H2 O
H2 O2
NAD
NADH
NAD
H2 O
NADH
H+
GSH
H2 O
NAD
NADH
H+
Acrolen
Cl-
NAD
H2 O
NADH
H+
Heme
Heme
Heme
Zinc
Excre
Cytosol
Hepatocyte
Endoplasmic Reticulum
Intestinal Epithelial Cell
Endoplasmic Reticulum
SLC22A1
ABCC3
CYP2C9
CYP3A4
CYP3A7
ALDH3A1
GSTA1
ADH1A
ALDH3A1
Cycloph
4GtyCP
chlogl
3DCLFA
4KcycPm
Nornm
Caroxyp
Alcopho
AcryliA
PhoAzdm
Phospho
Cycloph
Cycloph
Cycloph
Cycloph
Cycloph
Cycloph
Aldoph
Aldoph
AcryliA
PhoAzdm
Alcopho
4GtyCP
Nornm
3DCLFA
chlogl
4KcycPm
Phospho
Caroxyp
O2
NADPH
H+
4HCP
H2O
NADP
O2
H2O
H2O2
NAD
NADH
NAD
H2O
NADH
H+
GSH
H2O
NAD
NADH
H+
Acrolen
Cl
NAD
H2O
NADH
H+
Excre