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Cytochrome P450 3A4 Vildagliptin Vildagliptin Vildagliptin PIS1M1 Vildagliptin PIS1M1 Urinary Excretion and/or Bile duct Excretion Heme Hepatocytes Kidney Liver Cytosol Vildagliptin undergoes metabolism to give Vildagliptin PIS1M1. Endoplasmic Reticulum Bile Ducts Blood Vessel Blood Vessel
CYP3A4 Equa Equa Vil PIS Vil PIS U E a B Heme Hepatocytes Kidney Liver Cytosol Vildagliptin undergoes metabolism to give Vildagliptin PIS1M1. Endoplasmic Reticulum Bile Ducts Blood Vessel Blood Vessel
Endoplasmic Reticulum CYP3A4 Equa Equa Vil PIS Vil PIS U E a B