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Endoplasmic Reticulum Endoplasmic Reticulum Unknown Unknown Unknown CYP3A4 CYP3A4 CYP3A4 Tetrabenazine Tetrabenazine Tetrabenazine PIS1M2 Tetrabenazine PIS2M1 Tetrabenazine PIS2M1 Tetrabenazine PIS1M1 Tetrabenazine PIS1M2 Urinary Excretion and/or Bile duct Excretion