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Unknown Unknown Cytochrome P450 3A4 Cytochrome P450 3A4 Cytochrome P450 3A4 Fostamatinib Fostamatinib PIS4M1 Fostamatinib PIS4M1 Fostamatinib Fostamatinib PIS1M1 Fostamatinib PIS2M1 Heme Heme Heme Urinary Excretion and/or Bile duct Excretion Endoplasmic Reticulum Cytosol Hepatocyte Endoplasmic Reticulum Kidney Bile Ducts Liver Blood Vessel Blood Vessel Many other Cytochrome P450 enzymes are involved in Phase I (PI) Step 1(S1) and Step 2(S2) reactions. Fostamatinib undergoes metabolism to give Fostamatinib PIS1M1, Fostamatinib PIS2M1 and Fostamatinib PIS4M1.
Endoplasmic Reticulum Endoplasmic Reticulum Unknown Unknown CYP3A4 CYP3A4 CYP3A4 Fostamatinib Fostamatinib PIS4M1 Fostamatinib PIS4M1 Fostamatinib Fostamatinib PIS1M1 Fostamatinib PIS2M1 Urinary Excretion and/or Bile duct Excretion